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Novel urate transporter 1 (URAT1) inhibitors: a review of recent patent literature (2016?2019) 期刊论文
EXPERT OPINION ON THERAPEUTIC PATENTS, 2019, 卷号: 29, 期号: 11, 页码: 871-879
作者:  Dong, Yue;  Zhao, Tong;  Ai, Wei;  Zalloum, Waleed A.;  Kang, Dongwei
收藏  |  浏览/下载:11/0  |  提交时间:2019/12/11
Systematic Structure-Activity Relationship (SAR) Exploration of Diarylmethane Backbone and Discovery of A Highly Potent Novel Uric Acid Transporter 1 (URAT1) Inhibitor 期刊论文
MOLECULES, 2018, 卷号: 23, 期号: 2
作者:  Cai, Wenqing;  Wu, Jingwei;  Liu, Wei;  Xie, Yafei;  Liu, Yuqiang
收藏  |  浏览/下载:12/0  |  提交时间:2019/12/11
Synthesis, Crystal Structure and URAT1 Inhibitory Activity of 2-((5-Bromo-4-((4-cyclobutylnaphth-1-yl)methyl)-4H-1,2,4-triazol-3-yl)th io)acetic Acid 期刊论文
结构化学, 2017, 卷号: 36, 期号: 9, 页码: 1425-1432
作者:  Zhang Xiansheng;  Xin Xiao;  Liu Wei;  Xie Yafei;  Liu Changying
收藏  |  浏览/下载:6/0  |  提交时间:2019/12/16
The development of an effective synthetic route of lesinurad (RDEA594) 期刊论文
CHEMISTRY CENTRAL JOURNAL, 2017, 卷号: 11
作者:  Meng, Qing;  Zhao, Tong;  Kang, Dongwei;  Huang, Boshi;  Zhan, Peng
收藏  |  浏览/下载:10/0  |  提交时间:2019/12/12
Discovery of Flexible Naphthyltriazolylmethane-based Thioacetic Acids as Highly Active Uric Acid Transporter 1 (URAT1) Inhibitors for the Treatment of Hyperuricemia of Gout 期刊论文
MEDICINAL CHEMISTRY, 2017, 卷号: 13, 期号: 3, 页码: 260-281
作者:  Zhang, Xiansheng;  Wu, Jingwei;  Liu, Wei;  Liu, Yuqiang;  Xie, Yafei
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/12
Synthesis,Crystal Structure and URAT1 Inhibitory Activity of 2-((5-Bromo-4-((4-cyclobutylnaphth-1-yl)methyl)-4H-1,2,4-triazol-3-yl)thio)acetic Acid 期刊论文
结构化学, 2017, 期号: 09, 页码: 1425-1432
作者:  Zhang XS(张宪生);  Xin X(辛晓);  Liu W(刘巍);  Xie YF(谢亚非);  Liu ZY(刘长鹰)
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/12
Design, Synthesis and Biological Activity of Tetrazole-bearing Uric Acid Transporter 1 Inhibitors 期刊论文
高等学校化学研究, 2017, 卷号: 33, 期号: 1, 页码: 49-60
作者:  Cai Wenqing;  Liu Wei;  Xie Yafei;  Wu Jingwei;  Liu Yuqiang
收藏  |  浏览/下载:13/0  |  提交时间:2019/12/12
含大位阻结构的柔性尿酸转运体1(URAT1)抑制剂的设计、合成和生物活性研究 期刊论文
有机化学, 2017, 卷号: 37, 期号: 9, 页码: 2303-2314
作者:  蔡文卿;  刘巍;  张硕;  王建武;  赵桂龙
收藏  |  浏览/下载:8/0  |  提交时间:2019/12/12
痛风治疗新药——选择性尿酸重吸收抑制剂1esinurad 期刊论文
上海医药, 2016, 卷号: 37, 期号: 19
作者:  张炯;  刘磊;  薛愉;  杨雪;  梁敏锐
收藏  |  浏览/下载:13/0  |  提交时间:2019/12/05
Discovery of a Flexible Triazolylbutanoic Acid as a Highly Potent Uric Acid Transporter 1 (URAT1) Inhibitor 期刊论文
MOLECULES, 2016, 卷号: 21, 期号: 11
作者:  Tian, He;  Liu, Wei;  Zhou, Zhixing;  Shang, Qian;  Liu, Yuqiang
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/17


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