CORC

浏览/检索结果: 共14条,第1-10条 帮助

已选(0)清除 条数/页:   排序方式:
Design, Synthesis, and Biological Activities of Novel Triazolothiadiazole Derivatives Linked with Amino Side Chain Containing Urea Group as DOT1L Inhibitors 期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2020, 卷号: 40, 期号: 8, 页码: 2450-2459
作者:  Liu Na;  Guo Siqi;  Liu Junfang;  Chen Yantao;  Xu Xiaoming
收藏  |  浏览/下载:21/0  |  提交时间:2020/12/24
Structural Modifications of the Triazolo-thiadiazole Derivatives as DOT1L Inhibitors and Their Activities 期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2020, 卷号: 40, 期号: 5, 页码: 1345-1354
作者:  Xu Xiaoming;  Guo Siqi;  Zhang Jing;  Chen Yantao;  Kang Yaqing
收藏  |  浏览/下载:18/0  |  提交时间:2020/12/24
Lead discovery, chemical optimization, and biological evaluation studies of novel histone methyltransferase SET7 small-molecule inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 9, 页码: 10
作者:  Hou, Zeng;  Min, Wenjian;  Zhang, Rukang;  Niu, Ao;  Li, Yuanqing
收藏  |  浏览/下载:42/0  |  提交时间:2020/07/01
连氨基脲链的三氮唑并噻二唑类DOT1L抑制剂的设计、合成及活性 期刊论文
有机化学, 2020, 卷号: 40, 期号: 8, 页码: 2450
作者:  刘娜;  郭思岐;  刘俊芳;  陈彦韬;  徐晓明
收藏  |  浏览/下载:33/0  |  提交时间:2020/12/24
Design, synthesis and anti leukemia cells proliferation activities of pyrimidylaminoquinoline derivatives as DOT1L inhibitors 期刊论文
BIOORGANIC CHEMISTRY, 2018, 卷号: 80, 页码: 649-654
作者:  Zhang, Li;  Chen, Yantao;  Liu, Na;  Li, Linjuan;  Xiao, Senhao
收藏  |  浏览/下载:38/0  |  提交时间:2019/01/08
Discovery of potent DOT1L inhibitors by AlphaLISA based High Throughput Screening assay 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 8, 页码: 1751-1758
作者:  Song, Yakai;  Li, Linjuan;  Chen, Yantao;  Liu, Jingqiu;  Xiao, Senhao
收藏  |  浏览/下载:42/0  |  提交时间:2019/01/08
Convenient preparation of pinometostat and related 5 '-deoxy-5 '-amino adenosine derivatives as well as their activity against DOT1L 期刊论文
TETRAHEDRON LETTERS, 2018, 卷号: 59, 期号: 4, 页码: 415-417
作者:  Liu, Tongchao;  Ren, Huanming;  Li, Cong;  Chen, Guohua;  Cheng, Maosheng
收藏  |  浏览/下载:27/0  |  提交时间:2019/01/08
Inactivation of PBX3 and HOXA9 by down-regulating H3K79 methylation represses NPM1-mutated leukemic cell survival 期刊论文
THERANOSTICS, 2018, 卷号: 8, 期号: 16
作者:  Zhang, Wu;  Zhao, Chen;  Zhao, Junmei;  Zhu, Yongmei;  Weng, Xiangqin
收藏  |  浏览/下载:11/0  |  提交时间:2019/12/05
Preparation of 5 '-deoxy-5 '-amino-5 '-C-methyl adenosine derivatives and their activity against DOT1L 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 27, 期号: 22, 页码: 4960-4963
作者:  Liu, Tongchao;  Xie, Wuchen;  Li, Cong;  Ren, Huanming;  Mao, Yudong
收藏  |  浏览/下载:22/0  |  提交时间:2019/01/08
BET蛋白抑制剂I-BET151抗肝癌作用的表观遗传学机制研究 学位论文
2017, 2015
周仲实
收藏  |  浏览/下载:10/0  |  提交时间:2017/06/20


©版权所有 ©2017 CSpace - Powered by CSpace