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Design, synthesis, and biological evaluation of 4-benzoylamino-1H-pyrazole-3-carboxamide derivatives as potent CDK2 inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 215, 页码: 12
作者:  Lin, Tingting;  Li, Jiacheng;  Liu, Liping;  Li, Yuanqing;  Jiang, Hualiang
收藏  |  浏览/下载:70/0  |  提交时间:2021/05/24
Cediranib Induces Apoptosis, G1 Phase Cell Cycle Arrest, and Autophagy in Non-Small-Cell Lung Cancer Cell A549 In Vitro 期刊论文
BIOMED RESEARCH INTERNATIONAL, 2021, 卷号: 2021, 页码: 11
作者:  Guo, Menghuan;  Liu, Zhiyuan;  Si, Jing;  Zhang, Jinhua;  Zhao, Jin
收藏  |  浏览/下载:25/0  |  提交时间:2021/12/10
Design, synthesis, and molecular docking study of 3H-imidazole[4,5-c]pyridine derivatives as CDK2 inhibitors 期刊论文
ARCHIV DER PHARMAZIE, 2018, 卷号: 351, 期号: 6
作者:  Wu, Yi-Zhe;  Ying, Hua-Zhou;  Xu, Lei;  Cheng, Gang;  Chen, Jing
收藏  |  浏览/下载:31/0  |  提交时间:2019/01/08
Antitumor action of CDK inhibitor LS-007 as a single agent and in combination with ABT-199 against human acute leukemia cells 期刊论文
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 11, 页码: 1481-1489
作者:  Xie, Shao;  Jiang, Hui;  Zhai, Xiao-wen;  Wei, Fan;  Wang, Shu-dong
收藏  |  浏览/下载:25/0  |  提交时间:2019/01/08
Multiple CDK inhibitor dinaciclib suppresses neuroblastoma growth via inhibiting CDK2 and CDK9 activity 期刊论文
SCIENTIFIC REPORTS, 2016, 卷号: 6, 页码: 29090
作者:  Chen, Zhenghu;  Wang, Zhenyu;  Pang, Jonathan C;  Yu, Yang;  Bieerkehazhi, Shayahati
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/03
Multiple CDK inhibitor dinaciclib suppresses neuroblastoma growth via inhibiting CDK2 and CDK9 activity 期刊论文
SCIENTIFIC REPORTS, 2016, 卷号: 6
作者:  Chen, Zhenghu;  Wang, Zhenyu;  Pang, Jonathan C.;  Yu, Yang;  Bieerkehazhi, Shayahati
收藏  |  浏览/下载:2/0  |  提交时间:2019/12/06
ERK/GSK3β signaling is involved in atractylenolide I-induced apoptosis and cell cycle arrest in melanoma cells 期刊论文
Oncology reports, 2015, 卷号: 34, 期号: 3, 页码: 1543-8
作者:  Ye, Yan;  Chao, Xiao-Juan;  Wu, Jin-Feng;  Cheng, Brian Chi-Yan;  Su, Tao
收藏  |  浏览/下载:15/0  |  提交时间:2019/01/08
A new arylbenzofuran derivative functions as an anti-tumour agent by inducing DNA damage and inhibiting PARP activity 期刊论文
SCIENTIFIC REPORTS, 2015, 卷号: 5
作者:  Chen, Hongbo;  Zeng, Xiaobin;  Gao, Chunmei;  Ming, Pinghong;  Zhang, Jianping
收藏  |  浏览/下载:23/0  |  提交时间:2019/01/08
In Silico Identification and In Vitro and In Vivo Validation of Anti-Psychotic Drug Fluspirilene as a Potential CDK2 Inhibitor and a Candidate Anti-Cancer Drug 期刊论文
PLOS ONE, 2015, 卷号: 10, 期号: 7
作者:  Shi, Xi-Nan;  Li, Hongjian;  Yao, Hong;  Liu, Xu;  Li, Ling
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/04
Design, synthesis and biological evaluation of thienopyridinones as Chk1 inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2014, 卷号: 22, 期号: 17, 页码: 4882-4892
作者:  Song, Pinrao;  Peng, Peng;  Han, Mengmeng;  Cao, Xianchao;  Ma, Xiaodong
收藏  |  浏览/下载:22/0  |  提交时间:2019/01/08


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