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LS-106, a novel EGFR inhibitor targeting C797S, exhibits antitumor activities both in vitro and in vivo 期刊论文
CANCER SCIENCE, 2021, 页码: 12
作者:  Liu, Yingqiang;  Lai, Mengzhen;  Li, Shan;  Wang, Yanan;  Feng, Fang
收藏  |  浏览/下载:62/0  |  提交时间:2022/01/18
Design, synthesis and biological evaluation of potent EGFR kinase inhibitors against 19D/T790M/C797S mutation 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 16, 页码: 6
作者:  Su, Zhicheng;  Yang, Tingyuan;  Wang, Jie;  Lai, Mengzhen;  Tong, Linjiang
收藏  |  浏览/下载:27/0  |  提交时间:2020/12/24
EGFR  NSCLC  C797S  
2-Oxo-3,4-dihydropyrimido[4,5-d] pyrimidines as new reversible inhibitors of EGFR C797S (Cys797 to Ser797) mutant 期刊论文
CHINESE CHEMICAL LETTERS, 2020, 卷号: 31, 期号: 5, 页码: 1281-1287
作者:  Hu, Xianglong;  Xun, Qiuju;  Zhang, Tao;  Zhu, Su-Jie;  Li, Qian
收藏  |  浏览/下载:46/0  |  提交时间:2020/07/01
Discovery of N-(4-(6-Acetamidopyrimidin-4-yloxy)phenyl)-2-(2-(trifluoromethyl)phenyl)acetamide (CHMFL-FLT3-335) as a Potent FMS-like Tyrosine Kinase 3 Internal Tandem Duplication (FLT3-ITD) Mutant Selective Inhibitor for Acute Myeloid Leukemia 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 2, 页码: 875-892
作者:  Liang, Xiaofei;  Wang, Beilei;  Chen, Cheng;  Wang, Aoli;  Hu, Chen
收藏  |  浏览/下载:19/0  |  提交时间:2020/05/21
Comparative profiling of sarcoplasmic phosphoproteins in ovine muscle with different color stability 期刊论文
Food Chemistry, 2018, 卷号: 240, 页码: 104-111
作者:  Li, Meng;  Li, Zheng;  Li, Xin;  Xin, Jianzeng;  Wang, Ying
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/23
Evaluation of in vitro and in vivo activity of a multityrosine kinase inhibitor, AL3810, against human thyroid cancer 期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 11, 页码: 1533-1542
作者:  Xie, Qin;  Chen, Hui;  Ai, Jing;  Gao, Ying-lei;  Geng, Mei-yu
收藏  |  浏览/下载:17/0  |  提交时间:2019/01/08
Synthesis and structure-activity relationship study of pyrazolo[3,4-d]pyrimidines as tyrosine kinase RET inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 27, 期号: 11, 页码: 2544-2548
作者:  Wang, Chengyan;  Liu, Hongchun;  Song, Zilan;  Ji, Yinchun;  Xing, Li
收藏  |  浏览/下载:31/0  |  提交时间:2019/01/08
evaluationofinvitroandinvivoactivityofamultityrosinekinaseinhibitoral3810againsthumanthyroidcancer 期刊论文
actapharmacologicasinica, 2017, 卷号: 38, 期号: 11, 页码: 1533
作者:  Xie Qin;  Chen Hui;  Al Jing;  Gao Yinglei;  Geng Meiyu
收藏  |  浏览/下载:9/0  |  提交时间:2020/07/01
Necrotic pyknosis is a morphologically and biochemically distinct event from apoptotic pyknosis 期刊论文
JOURNAL OF CELL SCIENCE, 2016
Hou, Lin; Liu, Kai; Li, Yuhong; Ma, Shuang; Ji, Xunming; Liu, Lei
收藏  |  浏览/下载:3/0  |  提交时间:2017/12/04
Xijiao Dihuang Decoction combined with Yinqiao Powder reverses influenza virus-induced F-actin reorganization in PMVECs by inhibiting ERM phosphorylation 期刊论文
Journal of Traditional Chinese Medical Sciences, 2016, 卷号: 3, 期号: 1
作者:  Xuan Z., Wu Y., Zhang C., Zhang S., Chen X., Li S., Hao Y., Wang Q., Wang X., Zhang S.
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/06


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