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4-Oxo-1,4-dihydroquinoline-3-carboxamide Derivatives as New Axl Kinase Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 14, 页码: 6807-6825
Tan, Li; Zhang, Zhang; Gao, Dongylin; Luo, Jinfeng; Tu, Zheng-Chao; Li, Zhengqiu; Peng, Lijie; Ren, Xiaomei; Ding, Ke
收藏  |  浏览/下载:23/0  |  提交时间:2016/12/16
Combined inhibition of DDR1 and Notch signaling is a therapeutic strategy for KRAS-driven lung adenocarcinoma 期刊论文
NATURE MEDICINE, 2016, 卷号: 22, 期号: 3, 页码: 270-277
Ambrogio, Chiara; Gomez-Lopez, Gonzalo; Falcone, Mattia; Vidal, August; Nadal, Ernest; Crosetto, Nicola; Blasco, Rafael B.; Fernandez-Marcos, Pablo J.; Sanchez-Cespedes, Montserrat; Ren, Xiaomei; Wang, Zhen; Ding, Ke; Hidalgo, Manuel; Serrano, Manuel; Villanueva, Alberto; Santamaria, David; Barbacid, Mariano
收藏  |  浏览/下载:32/0  |  提交时间:2016/12/16
Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
Wang, Zhen; Bian, Huan; Bartual, Sergio G.; Du, Wenting; Luo, Jinfeng; Zhao, Hu; Zhang, Shasha; Mo, Cheng; Zhou, Yang; Xu, Yong; Tu, Zhengchao; Ren, Xiaomei; Lu, Xiaoyun; Brekken, Rolf A.; Yao, Libo; Bullock, Alex N.; Su, Jin; Ding, Ke
收藏  |  浏览/下载:51/0  |  提交时间:2016/12/16
GZD856, a novel potent PDGFR alpha/beta inhibitor, suppresses the growth and migration of lung cancer cells in vitro and in vivo 期刊论文
CANCER LETTERS, 2016, 卷号: 375, 期号: 1, 页码: 172-178
作者:  Song, Liyan;  Pang, Hongwen;  Ding, Ke;  Yu, Rongmin;  Zhang, Zhang
收藏  |  浏览/下载:21/0  |  提交时间:2018/12/13
Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
作者:  Yao, Libo;  Ding, Ke;  Su, Jin;  Bullock, Alex N.;  Brekken, Rolf A.
收藏  |  浏览/下载:33/0  |  提交时间:2018/12/13
4-Oxo-1,4-dihydroquinoline-3-carboxamide Derivatives as New Axl Kinase Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 14, 页码: 6807-6825
作者:  Tan, Li;  Zhang, Zhang;  Gao, Dongylin;  Luo, Jinfeng;  Tu, Zheng-Chao
收藏  |  浏览/下载:19/0  |  提交时间:2018/12/13
Combined inhibition of DDR1 and Notch signaling is a therapeutic strategy for KRAS-driven lung adenocarcinoma 期刊论文
NATURE MEDICINE, 2016, 卷号: 22, 期号: 3, 页码: 270-277
作者:  Villanueva, Alberto;  Santamaria, David;  Barbacid, Mariano;  Nadal, Ernest;  Crosetto, Nicola
收藏  |  浏览/下载:25/0  |  提交时间:2018/12/13
GZD856, a novel potent PDGFR alpha/beta inhibitor, suppresses the growth and migration of lung cancer cells in vitro and in vivo 期刊论文
CANCER LETTERS, 2016, 卷号: 375, 期号: 1, 页码: 172-178
Zhang, Zhang; Ren, Xiaomei; Lu, Xiaoyun; Wang, Deping; Hu, Xianjing; Zheng, Yi; Song, Liyan; Pang, Hongwen; Yu, Rongmin; Ding, Ke
收藏  |  浏览/下载:37/0  |  提交时间:2016/12/16
Small-Molecule BET Inhibitors in Clinical and Preclinical Development and Their Therapeutic Potential 期刊论文
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2015, 卷号: 15, 期号: 8, 页码: 776-794
Yu, Lei; Wang, Zhen; Zhang, Zhang; Ren, Xiaomei; Lu, Xiaoyun; Ding, Ke
收藏  |  浏览/下载:25/0  |  提交时间:2016/12/16
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M) 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
Chan, Shingpan; Han, Kun; Qu, Rong; Tong, Linjiang; Li, Yingjun; Zhang, Zhang; Cheng, Huimin; Lu, Xiaoyun; Patterson, Adam; Smaill, Jeff; Ren, Xiaomei; Ding, Jian; Xie, Hua; Ding, Ke
收藏  |  浏览/下载:246/0  |  提交时间:2016/12/16


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