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Covalent Inhibitors Allosterically Block the Activation of Rho Family Proteins and Suppress Cancer Cell Invasion 期刊论文
ADVANCED SCIENCE, 2020, 页码: 13
作者:  Sun, Zhongya;  Zhang, Hao;  Zhang, Yuanyuan;  Liao, Liping;  Zhou, Wen
收藏  |  浏览/下载:107/0  |  提交时间:2020/07/01
A Small-Molecule Inhibitor Targeting TRIP13 Suppresses Multiple Myeloma Progression 期刊论文
CANCER RESEARCH, 2020, 卷号: 80, 期号: 3, 页码: 536-548
作者:  Wang, Yingcong;  Huang, Jing;  Li, Bo;  Xue, Han;  Tricot, Guido
收藏  |  浏览/下载:54/0  |  提交时间:2020/07/01
Discovery and biological evaluation of vinylsulfonamide derivatives as highly potent, covalent TEAD autopalmitoylation inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 184, 页码: 15
作者:  Lu, Wenchao;  Wang, Jun;  Li, Yong;  Tao, Hongru;  Xiong, Huan
收藏  |  浏览/下载:96/0  |  提交时间:2020/07/01
Discovery of alkoxy benzamide derivatives as novel BPTF bromodomain inhibitors via structure-based virtual screening 期刊论文
BIOORGANIC CHEMISTRY, 2019, 卷号: 86, 页码: 494-500
作者:  Zhang, Dan;  Han, Jie;  Lu, Wenchao;  Lian, Fulin;  Wang, Jun
收藏  |  浏览/下载:11/0  |  提交时间:2020/07/01
Small-Molecule Targeting of Oncogenic FTO Demethylase in Acute Myeloid Leukemia 期刊论文
CANCER CELL, 2019, 卷号: 35, 期号: 4, 页码: 677-+
作者:  Huang, Yue;  Su, Rui;  Sheng, Yue;  Dong, Lei;  Dong, Ze
收藏  |  浏览/下载:26/0  |  提交时间:2020/07/01
The identification of novel small-molecule inhibitors targeting WDR5-MLL1 interaction through fluorescence polarization based high-throughput screening 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 4, 页码: 638-645
作者:  Ye, Xiaoqing;  Zhang, Rukang;  Lian, Fulin;  Zhang, Weiyao;  Lu, Wenchao
收藏  |  浏览/下载:4/0  |  提交时间:2020/07/01
Fragment-based drug discovery of triazole inhibitors to block PDE delta-RAS protein-protein interaction 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 163, 页码: 597-609
作者:  Chen, Danqi;  Chen, Yuehong;  Lian, Fulin;  Chen, Liu;  Li, Yanlian
收藏  |  浏览/下载:18/0  |  提交时间:2020/07/01
Fragment-based drug discovery of triazole inhibitors to block PDEδ-RAS protein-protein interaction 期刊论文
European journal of medicinal chemistry, 2018, 卷号: 163, 页码: 597-609
作者:  Chen, Danqi;  Chen, Yuehong;  Lian, Fulin;  Chen, Liu;  Li, Yanlian
收藏  |  浏览/下载:92/0  |  提交时间:2019/01/08
Pharmacological inhibition of dihydroorotate dehydrogenase induces apoptosis and differentiation in acute myeloid leukemia cells 期刊论文
HAEMATOLOGICA, 2018, 卷号: 103, 期号: 9, 页码: 1472-1483
作者:  Wu, Dang;  Wang, Wanyan;  Chen, Wuyan;  Lian, Fulin;  Lang, Li
收藏  |  浏览/下载:37/0  |  提交时间:2019/01/08
Discovery of 1,8-acridinedione derivatives as novel GCN5 inhibitors via high throughput screening 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 151, 页码: 740-751
作者:  Xiong, Huan;  Han, Jie;  Wang, Jun;  Lu, Wenchao;  Wang, Chen
收藏  |  浏览/下载:29/0  |  提交时间:2019/01/08


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