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科研机构
上海药物研究所 [13]
内容类型
期刊论文 [13]
发表日期
2021 [13]
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发表日期:2021
专题:上海药物研究所
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GPR84 signaling promotes intestinal mucosal inflammation via enhancing NLRP3 inflammasome activation in macrophages
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:
Zhang, Qing
;
Chen, Lin-hai
;
Yang, Hui
;
Fang, You-chen
;
Wang, Si-wei
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2022/01/18
GPR84
medium chain fatty acid receptor
GPCR
inflammatory bowel diseases
ulcerative colitis
NLRP3 inflammasome
macrophages
Sesquiterpenes from Artemisia Sieversiana and their anti-inflammatory activities
期刊论文
FITOTERAPIA, 2021, 卷号: 154, 页码: 7
作者:
Nuermaimaiti, Muaitaer
;
Turak, Ablajan
;
Yang, Qing
;
Tang, Bixi
;
Zang, Yi
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2021/11/04
Artemisia sieversiana
Dimeric guaianolides
Sesquiterpenes
Anti-inflammatory
Discovery of potential small molecular SARS-CoV-2 entry blockers targeting the spike protein
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 9
作者:
Wang, Lin
;
Wu, Yan
;
Yao, Sheng
;
Ge, Huan
;
Zhu, Ya
收藏
  |  
浏览/下载:86/0
  |  
提交时间:2021/11/04
SARS-CoV-2
natural products
virtual screening
spike protein
protein-protein interaction modulators
Triptolide analog LLDT-8 ameliorates psoriasis-like dermatitis in BALB/c mice via suppressing the IL-36 alpha signaling pathway
期刊论文
PHARMACOLOGICAL RESEARCH, 2021, 卷号: 169, 页码: 11
作者:
Qi, Qing
;
Li, Qian
;
Zhu, Hongwen
;
Lu, Huimin
;
Yang, Xiaoqian
收藏
  |  
浏览/下载:69/0
  |  
提交时间:2021/08/17
Triptolide
LLDT-8
Psoriasis
IL-36 alpha
IL-36 alpha pathway
Inflammation
Honokiol: A naturally occurring lignan with pleiotropic bioactivities
期刊论文
CHINESE JOURNAL OF NATURAL MEDICINES, 2021, 卷号: 19, 期号: 7, 页码: 481-490
作者:
Chen Cheng
;
Zhang Qing-Wen
;
Ye Yang
;
Lin Li-Gen
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2021/08/17
Honokiol
Natural sources
Ethnopharmacological uses
Physicochemical properties
Bioactivities
Clinical trials
Molecular insights into ago-allosteric modulation of the human glucagon-like peptide-1 receptor
期刊论文
NATURE COMMUNICATIONS, 2021, 卷号: 12, 期号: 1, 页码: 11
作者:
Cong, Zhaotong
;
Chen, Li-Nan
;
Ma, Honglei
;
Zhou, Qingtong
;
Zou, Xinyu
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2021/08/17
Design, synthesis and pharmacological evaluation of tricyclic derivatives as selective RXFP4 agonists
期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 110, 页码: 17
作者:
Lin, Lin
;
Lin, Guangyao
;
Zhou, Qingtong
;
Bathgate, Ross A. D.
;
Gong, Grace Qun
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2021/08/17
Synthesis
Structure-activity relationship
Relaxin family peptide receptor 4
Selective agonist
Molecular docking
Pharmacokinetics-based identification of pseudoaldosterogenic compounds originating from Glycyrrhiza uralensis roots (Gancao) after dosing LianhuaQingwen capsule
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 18
作者:
Lan, Xiao-fang
;
Olaleye, Olajide E.
;
Lu, Jun-lan
;
Yang, Wei
;
Du, Fei-fei
收藏
  |  
浏览/下载:75/0
  |  
提交时间:2021/06/11
LianhuaQingwen
glycyrrhetic acid
24-hydroxyglycyrrhetic acid
Gancao-induced pseudoaldosteronism
licorice-induced pseudoaldosteronism
11β
-hydroxysteroid dehydrogenase 2
COVID-19
colonic microbiota
Synthesis and Structure-Activity Relationships of Ring-Opened Bengamide Analogues against Methicillin-Resistant Staphylococcus aureus(dagger)
期刊论文
CHINESE JOURNAL OF CHEMISTRY, 2021, 卷号: 39, 期号: 3, 页码: 671-676
作者:
Yu, Chen-Xi
;
Wei, Bing-Yan
;
Kong, Xue-Qing
;
Yang, Cai-Guang
;
Nan, Fa-Jun
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2021/05/24
Bengamides
Staphylococcus aureus
Antibiotics
Structure‐
activity relationships
Pharmacokinetic
W2476 represses TXNIP transcription via dephosphorylation of FOXO1 at Ser319
期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2021, 页码: 11
作者:
Zhong, Li
;
Liu, Qing
;
Liu, Qiaofeng
;
Zhang, Shikai
;
Cao, Yongbing
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2021/05/24
chromatin immunoprecipitation
diabetes
transcription
TXNIP
W2476
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