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科研机构
安徽大学 [3]
合肥物质科学研究院 [2]
武汉大学 [1]
内容类型
期刊论文 [6]
发表日期
2018 [6]
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Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants including T315I for chronic myeloid leukemia
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 160, 页码: 61-81
作者:
Liu, Xuesong
;
Wang, Beilei
;
Chen, Cheng
;
Jiang, Zongru
;
Hu, Chen
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/11
ABL kinase
Kinase inhibitor
ABL mutant
CML
Discovery of (S)-2-amino-N-(5-(6-chloro-5-(3-methylphenylsulfonamido)pyridin-3-yl)-4-methylthiazol-2-yl)-3-methylbutanamide (CHMFL-PI3KD-317) as a potent and selective phosphoinositide 3-kinase delta (PI3K delta) inhibitor
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 156, 页码: 831-846
作者:
Liang, Xiaofei
;
Li, Feng
;
Chen, Cheng
;
Jiang, Zongru
;
Wang, Aoli
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/12/10
PI3K delta
Kinase inhibitor
Acute myeloid leukemia
Structure-activity relationship
Discovery of (S)-2-amino-N-(5-(6-chloro-5-(3-methylphenylsulfonamido)pyridin-3-yl)-4-methylthiazol-2-yl)-3-methylbutanamide (CHMFL-PI3KD-317) as a potent and selective phosphoinositide 3-kinase delta (PI3Kδ) inhibitor
期刊论文
European Journal of Medicinal Chemistry, 2018, 卷号: Vol.156, 页码: 831-846
作者:
Zongru Jiang
;
Wenliang Wang
;
Fengming Zou
;
Jing Liu
;
Qingsong Liu
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2019/04/22
PI3Kδ
Kinase
inhibitor
Acute
myeloid
leukemia
Structure-activity
relationship
Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants including T315I for chronic myeloid leukemia
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: Vol.160, 页码: 61-81
作者:
Liu, Xiaochuan
;
Wang, Beilei
;
Wang, Junjie
;
Zhang, Yicong
;
Jiang, Zongru
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/04/24
ABL kinase
Kinase inhibitor
ABL mutant
CML
Discovery of -2-amino-N-pyridin-3-yl)-4-methylthiazol-2-yl)-3-methylbutanamide as a potent and selective phosphoinositide 3-kinase delta inhibitor
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: Vol.156, 页码: 831-846
作者:
Liu, Xiaochuan
;
Jiang, Zongru
;
Li, Feng
;
Hu, Zhenquan
;
Ge, Juan
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/04/24
PI3K
delta
Kinase
inhibitor
Acute
myeloid
leukemia
Structure-activity
relationship
Compressive stress-strain relation of recycled aggregate concrete under cyclic loading
期刊论文
Construction and Building Materials, 2018, 卷号: 193
作者:
Hu, Xiaobin
;
Lu, Qinwang
;
Xu, Zihao
;
Zhang, Wenliang
;
Cheng, Shanshan
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2019/12/05
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