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科研机构
山东大学 [4]
复旦大学上海医学院 [1]
河南大学 [1]
内容类型
期刊论文 [6]
发表日期
2016 [6]
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发表日期:2016
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Arylazolyl(azinyl)thioacetanilides. Part 20: Discovery of novel purinylthioacetanilides derivatives as potent HIV-1 NNRTIs via a structure-based bioisosterism approach
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 18, 页码: 4424-4433
作者:
Lu, Xueyi
;
Li, Xiao
;
Yang, Jiapei
;
Huang, Boshi
;
Kang, Dongwei
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/17
HIV-1
AIDS
NNRTIs
Purinylthioacetanilide
Anti-HIV activity
Drug
design
Bioisosterism
Design, Synthesis, and Evaluation of Thiophene[3,2-d]pyrimidine Derivatives as HIV-1 Non-nucleoside Reverse Transcriptase Inhibitors with Significantly Improved Drug Resistance Profiles
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 17, 页码: 7991-8007
作者:
Kang, Dongwei
;
Fang, Zengjun
;
Li, Zhenyu
;
Huang, Boshi
;
Zhang, Heng
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/17
Arylazolyl(azinyl)thioacetanilides: Part 19: Discovery of Novel Substituted Imidazo[4,5-b]pyridin-2-ylthioacetanilides as Potent HIV NNRTIs Via a Structure-based Bioisosterism Approach
期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2016, 卷号: 88, 期号: 2, 页码: 241-253
作者:
Li, Xiao
;
Huang, Boshi
;
Zhou, Zhongxia
;
Gao, Ping
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/17
antiviral activity
drug design
HIV
imidazo[4,5-b]pyridin-2-ylthioacetanilides
molecular modeling
NNRTIs
SAR
First discovery of novel 3-hydroxy-quinazoline-2,4(1H,3H)-diones as specific anti-vaccinia and adenovirus agents via 'privileged scaffold' refining approach
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 21, 页码: 5182-5186
作者:
Kang, Dongwei
;
Zhang, Heng
;
Zhou, Zhongxia
;
Huang, Boshi
;
Naesens, Lieve
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2019/12/17
Quinolinone
Vaccinia
Adenovirus
Click chemistry
High-throughput
screening
Juvenile Hormone Activates the Transcription of Cell-division-cycle 6 (Cdc6) for Polyploidy-dependent Insect Vitellogenesis and Oogenesis
期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2016, 卷号: 291, 期号: 10, 页码: 5418-5427
作者:
Wu, Zhongxia[1]
;
Guo, Wei[2]
;
Xie, Yingtian[3]
;
Zhou, Shutang[4]
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/12/23
DNA replication
gene regulation
insect
juvenile hormone (JH)
reproduction
Topical 5-aminolevulinic acid photodynamic therapy improved refractory acne conglobata and perifolliculitis capitis abscedens et suffodiens rather than hidradenitis suppurativa
期刊论文
JOURNAL OF INNOVATIVE OPTICAL HEALTH SCIENCES, 2016, 卷号: 9, 期号: 1
作者:
Zhang, Linglin
;
Wang, Peiru
;
Shi, Lei
;
Zhang, Guolong
;
Zhang, Yunfeng
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  |  
浏览/下载:6/0
  |  
提交时间:2019/12/06
Acne conglobata
perifolliculitis capitis abscedens et suffodiens
hidradenitis suppurativa
aminolevunilic acid
photodynamic therapy
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