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科研机构
山东大学 [11]
内容类型
期刊论文 [11]
发表日期
2016 [11]
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共11条,第1-10条
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发表日期:2016
专题:山东大学
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Novel leucine ureido derivatives as aminopeptidase N inhibitors. Design, synthesis and activity evaluation
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 108, 页码: 21-27
作者:
Ma, Chunhua
;
Cao, Jiangying
;
Liang, Xuewu
;
Huang, Yongxue
;
Wu, Ping
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2019/12/16
Aminopeptidase N
Inhibitors
Leucine ureido derivatives
Synthesis
Discovery of BC-01, a novel mutual prodrug (hybrid drug) of ubenimex and fluorouracil as anticancer agent
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 121, 页码: 649-657
作者:
Jiang, Yuqi
;
Li, Xiaoyang
;
Hou, Jinning
;
Huang, Yongxue
;
Jia, Yuping
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2019/12/16
CD13
Ubenimex
Mutual prodrug
Antitumor
Anti-metastasis
Liver cancer
Design, Synthesis, and Antitumor Evaluation of 4-Amino-(1H)-pyrazole Derivatives as JAKs Inhibitors
期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 7, 期号: 10, 页码: 950-955
作者:
Liang, Xuewu
;
Zang, Jie
;
Zhu, Mengyuan
;
Gao, Qianwen
;
Wang, Binghe
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/12/16
JAKs
Inhibitors
4-Amino-(1H)-pyrazole
Anticancer
Discovery of a novel chimeric ubenimex-gemcitabine with potent oral antitumor activity
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 22, 页码: 5787-5795
作者:
Jiang, Yuqi
;
Hou, Jinning
;
Li, Xiaoyang
;
Huang, Yongxue
;
Wang, Xuejian
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/12/16
CD13 inhibitor
Ubenimex
Gemcitabine (GEM)
Anti-angiogenesis
Anticancer
Design, synthesis and preliminary biological evaluation of 4-aminopyrazole derivatives as novel and potent JAKs inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 12, 页码: 2660-2672
作者:
Liang, Xuewu
;
Huang, Yongxue
;
Zang, Jie
;
Gao, Qianwen
;
Wang, Binghe
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2019/12/16
Inhibitors
JAKs
Kinase
4-Aminopyrazole
Discovery of Multi-target Anticancer Agents Based on HDAC Inhibitor MS-275 and 5-FU
期刊论文
MEDICINAL CHEMISTRY, 2016, 卷号: 12, 期号: 1, 页码: 30-36
作者:
Jiang, Yuqi
;
Li, Xiaoguang
;
Li, Xiaoyang
;
Hou, Jinning
;
Ding, Yongzheng
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/12/16
Anticancer
HDAC
MS-275
Multitarget
5-Fluorouracil
Design, synthesis, and biological characterization of tamibarotene analogs as anticancer agents
期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2016, 卷号: 88, 期号: 4, 页码: 542-555
作者:
Jiang, Yuqi
;
Li, Xiaoyang
;
Wang, Xue
;
Wang, Zhonglan
;
Zhang, Jian
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/12/16
anticancer
histone deacetylases
multitarget drugs
retinoids
tamibarotene
PXD101 analogs with L-phenylglycine-containing branched cap as histone deacetylase inhibitors
期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2016, 卷号: 88, 期号: 4, 页码: 574-584
作者:
Li, Jingyao
;
Li, Xiaoyang
;
Wang, Xue
;
Hou, Jinning
;
Zang, Jie
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/12/16
antiproliferative activity
HDAC inhibitory activity
HDAC isoform
selectivity
HDACs
inhibitor
Design, Synthesis and Biological Evaluation of Novel Tamibarotene Derivative as Multitarget Anticancer Agent
期刊论文
Letters in Drug Design & Discovery, 2016, 卷号: 13, 期号: 8, 页码: 729-733
作者:
Jiang, Yuqi
;
Hou, Jinning
;
Li, Xiaoyang
;
Xu, Wenfang
;
Zhang, Yingjie
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2019/12/16
Tamibarotene (AM80)
multitarget
5-fluorouracil (5-FU)
anticancer
leukemia
Sohlh2 suppresses epithelial to mesenchymal transition in breast cancer via downregulation of IL-8
期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 31, 页码: 49411-49424
作者:
Ji, Shufang
;
Zhang, Wenfang
;
Zhang, Xiaoli
;
Hao, Chunyan
;
Hao, Aijun
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/17
Sohlh2
IL-8
EMT
metastasis
breast cancer
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