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Novel leucine ureido derivatives as aminopeptidase N inhibitors. Design, synthesis and activity evaluation 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 108, 页码: 21-27
作者:  Ma, Chunhua;  Cao, Jiangying;  Liang, Xuewu;  Huang, Yongxue;  Wu, Ping
收藏  |  浏览/下载:10/0  |  提交时间:2019/12/16
Discovery of BC-01, a novel mutual prodrug (hybrid drug) of ubenimex and fluorouracil as anticancer agent 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 121, 页码: 649-657
作者:  Jiang, Yuqi;  Li, Xiaoyang;  Hou, Jinning;  Huang, Yongxue;  Jia, Yuping
收藏  |  浏览/下载:8/0  |  提交时间:2019/12/16
Design, Synthesis, and Antitumor Evaluation of 4-Amino-(1H)-pyrazole Derivatives as JAKs Inhibitors 期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 7, 期号: 10, 页码: 950-955
作者:  Liang, Xuewu;  Zang, Jie;  Zhu, Mengyuan;  Gao, Qianwen;  Wang, Binghe
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/16
Discovery of a novel chimeric ubenimex-gemcitabine with potent oral antitumor activity 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 22, 页码: 5787-5795
作者:  Jiang, Yuqi;  Hou, Jinning;  Li, Xiaoyang;  Huang, Yongxue;  Wang, Xuejian
收藏  |  浏览/下载:2/0  |  提交时间:2019/12/16
Design, synthesis and preliminary biological evaluation of 4-aminopyrazole derivatives as novel and potent JAKs inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 12, 页码: 2660-2672
作者:  Liang, Xuewu;  Huang, Yongxue;  Zang, Jie;  Gao, Qianwen;  Wang, Binghe
收藏  |  浏览/下载:1/0  |  提交时间:2019/12/16
Discovery of Multi-target Anticancer Agents Based on HDAC Inhibitor MS-275 and 5-FU 期刊论文
MEDICINAL CHEMISTRY, 2016, 卷号: 12, 期号: 1, 页码: 30-36
作者:  Jiang, Yuqi;  Li, Xiaoguang;  Li, Xiaoyang;  Hou, Jinning;  Ding, Yongzheng
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/16
Design, synthesis, and biological characterization of tamibarotene analogs as anticancer agents 期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2016, 卷号: 88, 期号: 4, 页码: 542-555
作者:  Jiang, Yuqi;  Li, Xiaoyang;  Wang, Xue;  Wang, Zhonglan;  Zhang, Jian
收藏  |  浏览/下载:2/0  |  提交时间:2019/12/16
PXD101 analogs with L-phenylglycine-containing branched cap as histone deacetylase inhibitors 期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2016, 卷号: 88, 期号: 4, 页码: 574-584
作者:  Li, Jingyao;  Li, Xiaoyang;  Wang, Xue;  Hou, Jinning;  Zang, Jie
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/16
Design, Synthesis and Biological Evaluation of Novel Tamibarotene Derivative as Multitarget Anticancer Agent 期刊论文
Letters in Drug Design & Discovery, 2016, 卷号: 13, 期号: 8, 页码: 729-733
作者:  Jiang, Yuqi;  Hou, Jinning;  Li, Xiaoyang;  Xu, Wenfang;  Zhang, Yingjie
收藏  |  浏览/下载:6/0  |  提交时间:2019/12/16
Sohlh2 suppresses epithelial to mesenchymal transition in breast cancer via downregulation of IL-8 期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 31, 页码: 49411-49424
作者:  Ji, Shufang;  Zhang, Wenfang;  Zhang, Xiaoli;  Hao, Chunyan;  Hao, Aijun
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/17


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