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Mitochondrial Uncoupling Coordinated With PDH Activation Safely Ameliorates Hyperglycemia via Promoting Glucose Oxidation 期刊论文
DIABETES, 2019, 卷号: 68, 期号: 12, 页码: 2197-2209
作者:  Jiang, Haowen;  Jin, Jia;  Duan, Yanan;  Xie, Zhifu;  Li, Yufeng
收藏  |  浏览/下载:24/0  |  提交时间:2020/07/01
Natural Product Albiziabioside A Conjugated with Pyruvate Dehydrogenase Kinase Inhibitor Dichloroacetate To Induce Apoptosis-Ferroptosis-M2-TAMs Polarization for Combined Cancer Therapy 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 19, 页码: 8760-8772
作者:  Wei, Gaofei;  Sung, Jiahong;  Luan, Weijing;  Hou, Zhuang;  Wang, Shuai
收藏  |  浏览/下载:18/0  |  提交时间:2020/07/01
Switching off IMMP2L signaling drives senescence via simultaneous metabolic alteration and blockage of cell death 期刊论文
CELL RESEARCH, 2018, 卷号: 28, 期号: 6, 页码: 625-643
作者:  Yuan, Lifeng;  Zhai, Linhui;  Qian, Lili;  Huang, De;  Ding, Yi
收藏  |  浏览/下载:35/0  |  提交时间:2019/01/08
Development of the First Generation of Disulfide-Based Subtype Selective and Potent Covalent Pyruvate Dehydrogenase Kinase 1 (PDK1) Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 6, 页码: 2227-2244
作者:  Liu, Yifu;  Xie, Zuoquan;  Zhao, Dan;  Zhu, Jin;  Mao, Fei
收藏  |  浏览/下载:22/0  |  提交时间:2019/01/08
Mitochondrial uncoupling combined with pyruvate dehydrogenase activity ameliorated hyperglycaenia 会议论文
作者:  Jiang, H. -W.;  Li, J. -Y;  Xie, Z. -F.;  Gao, A. -H.;  Zhang, L. -N.
收藏  |  浏览/下载:8/0  |  提交时间:2019/01/08
miR-182 Regulates Metabolic Homeostasis by Modulating Glucose Utilization in Muscle 期刊论文
CELL REPORTS, 2016, 卷号: 16, 期号: 3, 页码: 757-768
作者:  Zhang, Duo;  Li, Yan;  Yao, Xuan;  Wang, Hui;  Zhao, Lei
收藏  |  浏览/下载:33/0  |  提交时间:2019/01/08
JX06 Selectively Inhibits Pyruvate Dehydrogenase Kinase PDK1 by a Covalent Cysteine Modification 期刊论文
CANCER RESEARCH, 2015, 卷号: 75, 期号: 22, 页码: 4923-4936
作者:  Sun, Wenyi;  Xie, Zuoquan;  Liu, Yifu;  Zhao, Dan;  Wu, Zhixiang
收藏  |  浏览/下载:29/0  |  提交时间:2019/01/08
Lactate Dehydrogenase B Is Associated with the Response to Neoadjuvant Chemotherapy in Oral Squamous Cell Carcinoma 期刊论文
PLOS ONE, 2015, 卷号: 10, 期号: 5
作者:  Sun, Wenyi;  Zhang, Xiaomin;  Ding, Xu;  Li, Huaiqi;  Geng, Meiyu
收藏  |  浏览/下载:17/0  |  提交时间:2019/01/08
丙酮酸脱氢酶激酶共价抑制剂JX06抗肿瘤活性和机制研究(英文) 会议论文
作者:  孙文怡;  谢作权;  刘逸夫;  赵丹;  武志翔
收藏  |  浏览/下载:29/0  |  提交时间:2019/01/08
JX06 selectively inhibits pyruvate dehydrogenase kinase 1 by covalently targeting a cysteine residue 会议论文
作者:  Sun WY(孙文怡);  Xie ZQ(谢作权);  Liu YF(刘逸夫);  Zhao D(赵丹);  Wu ZX(武志翔)
收藏  |  浏览/下载:15/0  |  提交时间:2019/01/08


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