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科研机构
北京大学 [31]
内容类型
期刊论文 [31]
发表日期
2017 [4]
2016 [3]
2015 [3]
2014 [1]
2013 [2]
2011 [2]
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专题:北京大学
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Aldehyde dehydrogenase 1A1 increases NADH levels and promotes tumor growth via glutathione/dihydrolipoic acid-dependent NAD(+) reduction
期刊论文
ONCOTARGET, 2017
Wang, Baiyun
;
Chen, Xue
;
Wang, Zixi
;
Xiong, Wei
;
Xu, Tao
;
Zhao, Xinyuan
;
Cao, Yang
;
Guo, Yanru
;
Li, Lin
;
Chen, She
;
Huang, Song
;
Wang, Xiaodong
;
Fang, Min
;
Shen, Zhirong
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2017/12/03
aldehyde dehydrogenase
lung cancer
glutathione
dihydrolipoic acid
NAD(+)/NADH ratio
SELECTIVE INHIBITORS
OXIDATIVE STRESS
BREAST-CANCER
RETINOIC ACID
LUNG-CANCER
STEM-CELLS
VITAMIN-E
ALDH1A1
ALDH3A1
METABOLISM
Selective inhibition of Ebola entry with selective estrogen receptor modulators by disrupting the endolysosomal calcium
期刊论文
SCIENTIFIC REPORTS, 2017
Fan, Hanlu
;
Du, Xiaohong
;
Zhang, Jingyuan
;
Zheng, Han
;
Lu, Xiaohui
;
Wu, Qihui
;
Li, Haifeng
;
Wang, Han
;
Shi, Yi
;
Gao, George
;
Zhou, Zhuan
;
Tan, Dun-Xian
;
Li, Xiangdong
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/03
DRUG-INDUCED PHOSPHOLIPIDOSIS
NIEMANN-PICK C1
VIRUS GLYCOPROTEIN
FUNCTIONAL INHIBITORS
NPC1(+) ENDOLYSOSOMES
PLASMA-MEMBRANE
CELL ENTRY
FUSION
CHOLESTEROL
INFECTION
Discovery of a Highly Potent, Selective, and Metabolically Stable Inhibitor of Receptor-Interacting Protein 1 (RIP1) for the Treatment of Systemic Inflammatory Response Syndrome
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017
Ren, Yan
;
Su, Yaning
;
Sun, Liming
;
He, Sudan
;
Meng, Lingjun
;
Liao, Daohong
;
Liu, Xiao
;
Ma, Yongfen
;
Liu, Chunyan
;
Li, Sisi
;
Ruan, Hanying
;
Lei, Xiaoguang
;
Wang, Xiaodong
;
Zhang, Zhiyuan
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2017/12/03
EXPERIMENTAL DISEASE-MODELS
CELL-DEATH
KINASE INHIBITORS
INDUCED SHOCK
NECROPTOSIS
NECROSIS
NECROSTATIN-1
SPECIFICITY
INJURY
ALPHA
Rational Design of Selective Allosteric Inhibitors of PHGDH and Serine Synthesis with Anti-tumor Activity
期刊论文
CELL CHEMICAL BIOLOGY, 2017
Wang, Qian
;
Liberti, Maria V.
;
Liu, Pei
;
Deng, Xiaobing
;
Liu, Ying
;
Locasale, Jason W.
;
Lai, Luhua
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2017/12/03
PHOSPHOGLYCERATE DEHYDROGENASE
CANCER METABOLISM
SYNTHESIS PATHWAY
ACCURATE DOCKING
BINDING-SITES
DRUG DESIGN
BIOSYNTHESIS
DISCOVERY
CELLS
COMBINATION
Serotonin transporter polymorphism alters citalopram effects on human pain responses to physical pain
期刊论文
NEUROIMAGE, 2016
Ma, Yina
;
Wang, Chenbo
;
Luo, Siyang
;
Li, Bingfeng
;
Wager, Tor D.
;
Zhang, Wenxia
;
Rao, Yi
;
Han, Shihui
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2017/12/03
SSRI
5-HTTLPR
fMRI
Pain perception
Personalized medicine
HUMAN BRAIN
5-HTTLPR POLYMORPHISM
SUBJECTIVE EXPERIENCE
GENE POLYMORPHISM
INDIVIDUAL-DIFFERENCES
PROMOTER POLYMORPHISM
SOMATOSENSORY CORTEX
THERMAL HYPERALGESIA
NEURAL MECHANISMS
HEALTHY-SUBJECTS
Crosslinked Aspartic Acids as Helix-Nucleating Templates
期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2016
Zhao, Hui
;
Liu, Qi-Song
;
Geng, Hao
;
Tian, Yuan
;
Cheng, Min
;
Jiang, Yan-Hong
;
Xie, Ming-Sheng
;
Niu, Xiao-Gang
;
Jiang, Fan
;
Zhang, Ya-Ou
;
Lao, Yuan-Zhi
;
Wu, Yun-Dong
;
Xu, Nai-Han
;
Li, Zi-Gang
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2017/12/04
amino acids
circular dichroism
helical structures
peptides
protein-protein interactions
HYDROGEN-BOND SURROGATE
PROTEIN-PROTEIN INTERACTIONS
RECEPTOR-COACTIVATOR INTERACTIONS
SHORT ALPHA-HELICES
ESTROGEN-RECEPTOR
FORCE-FIELD
CYCLIC-PEPTIDES
CONFORMATIONAL-ANALYSIS
SELECTIVE INHIBITORS
STAPLED PEPTIDES
Discovery of Novel Polo-Like Kinase 1 Polo-Box Domain Inhibitors to Induce Mitotic Arrest in Tumor Cells
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016
Qin, Tan
;
Chen, Fangjin
;
Zhuo, Xiaolong
;
Guo, Xiao
;
Yun, Taikangxiang
;
Liu, Ying
;
Zhang, Chuanmao
;
Lai, Luhua
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2017/12/04
ADVANCED SOLID MALIGNANCIES
GROWTH IN-VIVO
PHASE-I
CELLULAR UPTAKE
PLK1
POLO-LIKE-KINASE-1
CANCER
PHOSPHOPEPTIDES
IDENTIFICATION
RECOGNITION
Muscarinic inhibition of nicotinic transmission in rat sympathetic neurons and adrenal chromaffin cells
期刊论文
PHILOSOPHICAL TRANSACTIONS OF THE ROYAL SOCIETY B-BIOLOGICAL SCIENCES, 2015
He, Lin-Ling
;
Zhang, Quan-Feng
;
Wang, Lie-Cheng
;
Dai, Jing-Xia
;
Wang, Chang-He
;
Zheng, Liang-Hong
;
Zhou, Zhuan
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2017/12/03
nAchRs
mAchRs
methacholine
nicotine
G-proteins
TRANSMITTER RELEASE
SYNAPTIC-TRANSMISSION
GANGLION NEURONS
DOPAMINE RELEASE
G-PROTEIN
ACETYLCHOLINE-RECEPTORS
CATECHOLAMINE SECRETION
AMPEROMETRIC DETECTION
PRESYNAPTIC RECEPTORS
QUANTAL SECRETION
Allelic variation in 5-HTTLPR and the effects of citalopram on the emotional neural network
期刊论文
2015
Ma Yina
;
Li Bingfeng
;
Wang Chenbo
;
Zhang Wenxia
;
Rao Yi
;
Han Shihui
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2015/11/13
Meclofenamic acid selectively inhibits FTO demethylation of m(6)A over ALKBH5
期刊论文
核酸研究, 2015
Huang, Yue
;
Yan, Jingli
;
Li, Qi
;
Li, Jiafei
;
Gong, Shouzhe
;
Zhou, Hu
;
Gan, Jianhua
;
Jiang, Hualiang
;
Jia, Gui-Fang
;
Luo, Cheng
;
Yang, Cai-Guang
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2015/11/15
PROMOTE PROTEIN STABILITY
OBESITY-ASSOCIATED FTO
OXIDATIVE DEMETHYLATION
CRYSTAL-STRUCTURES
RNA DEMETHYLASE
ALKYLATION DAMAGE
ESCHERICHIA-COLI
MESSENGER-RNA
HISTONE DEMETHYLASES
MAXIMUM-LIKELIHOOD
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