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科研机构
北京大学 [10]
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期刊论文 [10]
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2017 [1]
2016 [2]
2015 [2]
2014 [3]
2013 [1]
2012 [1]
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专题:北京大学
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Highly Selective Activation of Heat Shock Protein 70 by Allosteric Regulation Provides an Insight into Efficient Neuroinflammation Inhibition
期刊论文
EBIOMEDICINE, 2017
Wang, Li-Chao
;
Liao, Li-Xi
;
Lv, Hai-Ning
;
Liu, Dan
;
Dong, Wei
;
Zhu, Jian
;
Chen, Jin-Feng
;
Shi, Meng-Ling
;
Fu, Ge
;
Song, Xiao-Min
;
Jiang, Yong
;
Zeng, Ke-Wu
;
Tu, Peng-Fei
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/03
Heat shock protein 70 (Hsp70)
Handelin
Drug target
Covalent modification
Neuroinflammation
HEAT-SHOCK PROTEINS
T-CELL REGULATION
HIGH-FAT DIET
KAPPA-B
AUTOIMMUNE ARTHRITIS
HSP70
STRESS
INFLAMMATION
EXPRESSION
POLYUBIQUITINATION
Total flavonoid aglycones extract in Radix scutellariae inhibits lung carcinoma and lung metastasis by affecting cell cycle and DNA synthesis
期刊论文
JOURNAL OF ETHNOPHARMACOLOGY, 2016
Wang, Yang
;
Cao, Hui-juan
;
Sun, Shu-jun
;
Dai, Jian-ye
;
Fang, Jun-wei
;
Li, Qian-hua
;
Yan, Chao
;
Mao, Wen-wei
;
Zhang, Yong-yu
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/04
Total flavonoid aglycones extract
Lung carcinoma
Cell cycle
DNA synthesis
CANCER CELLS
IN-VITRO
PLANIPES
ARREST
Electrophoretic deposition of colloidal particles on Mg with cytocompatibility, antibacterial performance, and corrosion resistance
期刊论文
ACTA BIOMATERIALIA, 2016
Sun, Jiadi
;
Zhu, Ye
;
Meng, Long
;
Chen, Peng
;
Shi, Tiantian
;
Liu, Xiaoya
;
Zheng, Yufeng
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/04
Magnesium
Colloidal particles
EPD
Functional coating
Corrosion
BIODEGRADABLE MAGNESIUM ALLOYS
IMPLANTS APPLICATION
ORTHOPEDIC IMPLANTS
STAINLESS-STEEL
CELL-ADHESION
SURFACE
TITANIUM
BONE
COATINGS
ACID
Sangxingtang inhibits the inflammation of LPS-induced acute lung injury in mice by down-regulating the MAPK/NF-κB pathway
期刊论文
Chinese Journal of Natural Medicines, 2015
Zhang Tianzhu
;
Yang Shihai
;
Yao Jinfu
;
Du Juan
;
Yan Tianhua
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2017/12/04
Sangxingtang
Inflammation
LPS-induced acute lung injury
MAPK/NF-κB pathway
IN-VITRO
ENDOTOXEMIA
HEMORRHAGE
EXPRESSION
APIGENIN
ALPHA
CELLS
RATS
VIVO
Diverse Ways of Perturbing the Human Arachidonic Acid Metabolic Network To Control Inflammation
期刊论文
ACCOUNTS OF CHEMICAL RESEARCH, 2015
Meng, Hu
;
Liu, Ying
;
Lai, Luhua
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2017/12/03
PROSTAGLANDIN E-2 SYNTHASE-1
TRADITIONAL CHINESE MEDICINE
LEUKOTRIENE A(4) HYDROLASE
DUAL INHIBITORS
DRUG DESIGN
LTA(4) HYDROLASE
5-LIPOXYGENASE
DISCOVERY
DERIVATIVES
CYCLOOXYGENASE-2
A perylene derivative regulates HIF-1 alpha and Stat3 signaling pathways
期刊论文
生物有机化学与医药化学, 2014
Chen, Han
;
Guan, Yongli
;
Yuan, Gu
;
Zhang, Qiang
;
Jing, Naijie
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2015/11/10
Stat3: the signal transducer and activator of transcription 3
HIF-1 alpha: hypoxia-inducible factor-1 alpha
Pancreatic cancer therapy
Breast cancer therapy
TEL03: a dual inhibitor of HIF-1 alpha and Stat3
HYPOXIA-INDUCIBLE FACTOR-1
G-QUARTET OLIGONUCLEOTIDES
HUMAN ERYTHROPOIETIN GENE
HUMAN PANCREATIC-CANCER
PROSTATE-CANCER
TARGETING STAT3
BREAST-CANCER
TRANSCRIPTIONAL ACTIVATION
CONSTITUTIVE ACTIVATION
LIGAND AGGREGATION
Development of 3,5-dinitrobenzoate-based 5-lipoxygenase inhibitors
期刊论文
生物有机化学与医药化学, 2014
Shang, Erchang
;
Liu, Ying
;
Wu, Yiran
;
Zhu, Wei
;
He, Chong
;
Lai, Luhua
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2015/11/10
3,5-Dinitrobenzoate
5-Lipoxygenase inhibitors
Cell-free assay
Human whole blood assay
SAR study
DISEASE
BIOSYNTHESIS
LEUKOTRIENES
INFLAMMATION
EICOSANOIDS
MECHANISMS
The Effects of Morin on Lipopolysaccharide-Induced Acute Lung Injury by Suppressing the Lung NLRP3 Inflammasome
期刊论文
inflammation, 2014
Zhang Tianzhu
;
Yang Shihai
;
Du Juan
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2015/11/11
morin
NLRP3 inflammasome
LPS-induced acute lung injury
ENDOTOXEMIA
HEMORRHAGE
RESPONSES
ALPHA
Tailoring the pH Dependence of Human Non-pancreatic Secretory Phospholipase A(2) by Engineering Surface Charges
期刊论文
应用生物化学与生物技术, 2013
Qiu, Shunchen
;
Lai, Luhua
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2015/11/10
Phospholipase A(2)
Protein engineering
Enzyme reaction optimum pH
Catalytic mechanism
The catalytic triad mechanism
The calcium-coordinated oxyanion mechanism
GROUP-IIA
ACTIVE-SITE
CATALYTIC MECHANISM
SERINE-PROTEASE
PANCREATIC PHOSPHOLIPASE-A2
CRYSTAL-STRUCTURE
ENZYME CATALYSIS
OPTIMUM
BINDING
STABILITY
Dynamic Modeling of Human 5-Lipoxygenase-Inhibitor Interactions Helps To Discover Novel Inhibitors
期刊论文
journal of medicinal chemistry, 2012
Wu, Yiran
;
He, Chong
;
Gao, Yang
;
He, Shan
;
Liu, Ying
;
Lai, Luhua
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2015/11/13
PROSTAGLANDIN E-2 SYNTHASE-1
HUMAN WHOLE-BLOOD
3-DIMENSIONAL STRUCTURES
THERAPEUTIC TARGET
POTENT INHIBITORS
DUAL INHIBITORS
CYCLOOXYGENASE
BIOSYNTHESIS
INFLAMMATION
LICOFELONE
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