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New heteroaryl-substituted piperidine compounds are protease-activated receptor antagonists useful for the treatment and/or prophylaxis of e.g. cardiovascular diseases, thromboembolic diseases, tumors, stroke, hypertension and asthma 专利
作者:  Heimbach, Dirk, Dr., 40629 Düsseldorf, DE;  Röhrig, Susanne, Dr., 40724 Hilden, DE;  Schneider, Dirk, 42115 Wuppertal, DE;  Rester, Ulrich, Dr., 42115 Wuppertal, DE;  Bender, Eckhard, Dr., 40764 Langenfeld, DE
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The modified lysosomal disorders of the central nervous system for the treatment and prevention of fault and (3R, 4R, 5S) - 3, 4 - diol (difluoromethyl) piperidine -5 - regimen 专利
作者:  クラーク シーン
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N-OXIDES OF PYRIDYLMETHYLPIPERAZINE AND -PIPERIDINE DERIVATIVES 专利
作者:  VAN AAR Marcel P M;  VAN AMSTERDAM Peter H;  BARF Gerrit A;  BAKKER Johan Antoine;  DEN BESTEN Cathaline
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PIPERIDINE DERIVATIVE AND COMPOSITION FOR INHIBITING NICOTINAMIDE PHOSPHORIBOSYL TRANSFERASE 专利
作者:  KENNETH W BAIR;  TIMM BAUMEISTER;  ALEXANDRE J BUCKMELTER;  KARL H CLODFELTER;  HAN BINGSONG
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N-(5S, 6S, 9R)-5-AMINO-6-(2, 3-DIFLUOROPHENYL)-6, 7, 8, 9-TETRAHYDRO-5H-CYCLOHEPTA[B]PYRIDIN-9-YL-4-(2-OXO-2, 3-DIHYDRO-1H-IMIDAZO[4, 5-B]PYRIDIN-1-YL)PIPERIDINE-1-CARBOXYLATE SALT 专利
作者:  Daniel Richard Roberts;  Richard Raymond Schartman;  Chenkou Wei
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/05
SUBSTITUTED 4-ALKYL- AND 4-ALKANOYL-PIPERIDINE DERIVATIVES AND THEIR USE AS NEUROKININ ANTAGONISTS 专利
作者:  JANSSENS Frans Eduard;  SOMMEN François Maria;  DE BOECK Benoît Christian Albert Ghislain;  LEENAERTS Joseph Elisabeth
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N- (5S, 6S, 9R) - 5 -AMINO- 6 - (2, 3 - DIFLUOROPHENYL) -6, 7, 8, 9 - TETRAHYDRO - 5H - CYCLOHEPTA [B] PYRIDIN-9 -YL- 4 - (2 - OXO-2, 3 - DIHYDRO - 1H- IMIDAZO [4, 5 -B] PYRIDIN - 1 - YL) PIPERIDINE - 1 - CARBOXYLATE, HEMISULFATE SALT 专利
作者:  ROBERTS DANIEL RICHARD;  SCHARTMAN RICHARD RAYMOND;  WEI CHENKOU
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PIPERIDINE DERIVATIVES AS SUBTYPE SELECTIVE N-METHYL-D-ASPARTATE ANTAGONISTS 专利
作者:  KORNBERG, Brian, Edward;  LEWTHWAITE, Russell, Andrew;  MANNING, David, Douglas;  NIKAM, Sham, Shridhar;  SCOTT, Ian, Leslie
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4-BENZYL PIPERIDINE ALKYLSULFOXIDE HETEROCYCLES AND THEIR USE AS SUBTYPE-SELECTIVE NMDA RECEPTOR ANTAGONISTS 专利
作者:  WRIGHT JONATHAN L;  KESTEN SUZANNE ROSS;  UPASANI RAVINDRA B;  LAN NANCY C
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PIPERIDINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME AS ACTIVE INGREDIENT 专利
作者:  OCHIAI, HIROSHI;  NISHITA, YOSHITAKA;  OHTANI, TAZUMI;  HAMANO, MASAYA
收藏  |  浏览/下载:2/0  |  提交时间:2019/12/05


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