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Preparing bis-halogenated-phenyl-(1,3,5)-triazine compound, comprises e.g. performing addition reaction on halogenated benzonitrile in alcohol in the presence of sodium methoxide, and cyclizing the obtained benzamidine hydrochloride. 专利
申请日期: 2012-01-01, 公开日期: 2012-03-21
作者:  JIAN X LIU C LU D ZHANG S WANG J
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/18
As the inhibitor for the treatment of cancer of the protein kinase, 3-(indazol-5-yl)-(1, 2, 4) triazine derivative, and related compd. 专利
作者:  チャン, ティン-ヤウ;  フィッシュマン, ティエリー オー.;  マッコイ, マーク エー.;  マク キットリック, ブライアン;  プロンガイ, アンドリュー
收藏  |  浏览/下载:6/0  |  提交时间:2019/12/05
New 4-aminopyrazol-(1, 5-a)-1, 3, 5-triazine derivatives, are potent and selective phosphodiesterase 4 inhibitors useful e.g. for treating CNS disorders, neuroinflammation, Crohn' s disease, asthma, cancer or epilepsy 专利
作者:  BOURGUIGNON JEAN JACQUES;  LUGNIER CLAIRE;  SCHMITT MARTINE;  MATHIEU ROMAIN;  MACHER JEAN PAUL
收藏  |  浏览/下载:2/0  |  提交时间:2019/12/05
DERIVATIVES 4 (BENZYLIDENE) - 3- ([METILSULFANIL]) - 4H-1, 2, 4-TRIAZINE-5- IT, POSSESSING THE INHIBITING ACTION WITH RESPECT TO PHOSPHODIESTERASE IV and ANTAGONISTIC ACTION with respect to TNF, FOR TREATING OF HEART DISEASES and ALLERGY 专利
作者:  Ханс-Михаэль ЭГГЕНВАЙЛЕР (DE);  Михаэль ВОЛЬФ (DE);  Норберт БАЙЕР (DE);  Йоахим ЛАЙБРОКК (DE);  Пьер ШЕЛЛИНГ (DE)
收藏  |  浏览/下载:1/0  |  提交时间:2019/12/05
DERIVED FROM 3 (3, 5-DIOXO-4, 5-DIHYDRO-3H- (1, 2, 4) TRIAZINE-2-YL) - BENZAMIDE BEING USED As INHIBITORS OF P2X7 FOR the TREATMENT OF INFLAMMATORY DISEASES 专利
作者:  DOMBROSKI MARK ANTHONY;  DUPLANTIER ALLEN JACOB
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1, 3, 5 - TRIAZINE DERIVATIVES, COMPOSITIONS COMPRISING THEM AND USES THEREOF IN THE MANUFACTURE OF MEDICAMENTS FOR THE TREATMENT OF PARKINSON' S DISEASE 专利
作者:  null
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DERIVATIVES OF 1, 3, 5-TRIAZINE, PHARMACEUTICAL COMPOSITION BASED ON THEREOF AND THEIR USING 专利
作者:  DEN KHARTOG JAKOBUS A. DZH.;  REJNDERS JAN KH.;  VAN SKHARRENBJURG GJUSTAAF DZH. M.;  PRAS-RAVES MARIA L.;  GJUSTAFSON GARI R.
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