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上海药物研究所 [14]
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Virtual Screening for Type II B Inhibitors of B-Raf(V600E) Kinase
期刊论文
CURRENT COMPUTER-AIDED DRUG DESIGN, 2020
作者:
Qiu, Kai-Xiong
;
Zhang, Wen
;
Yu, Fang
;
Li, Wei
;
Sun, Zhong-Wen
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2021/01/05
Ensemble-based virtual screening in discovering potent inhibitors targeting Von Hippel-Lindau (VHL) E3 ubiquitin ligase
期刊论文
LIFE SCIENCES, 2020
作者:
Liu, Yi
;
Lei, Yu
;
Guo, Sheng
;
Zuo, Zhili
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2021/01/05
The discovery, design and synthesis of potent agonists of adenylyl cyclase type 2 by virtual screening combining biological evaluation
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020
作者:
Xu, Guowei
;
Yang, Yaqing
;
Yang, Yanming
;
Song, Gao
;
Li, Shanshan
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  |  
浏览/下载:22/0
  |  
提交时间:2021/01/05
The discovery of novel and selective fatty acid binding protein 4 inhibitors by virtual screening and biological evaluation
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 18, 页码: 4310-4317
作者:
Song, Ming
;
Xu, Yong
;
Zhang, Yan
;
Nie, Tao
;
Zhou, Yang
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2018/12/13
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
作者:
Tu, Zhengchao
;
Zhou, Yulai
;
Ding, Ke
;
Xu, Yong
;
Xue, Xiaoqian
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  |  
浏览/下载:25/0
  |  
提交时间:2018/12/13
Identification of N-phenyl-2-(N-phenylphenylsulfonamido) acetamides as new ROR gamma inverse agonists: Virtual screening, structure-based optimization, and biological evaluation
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 116, 页码: 13-26
作者:
Xue, Xiaoqian
;
Song, Yu
;
Qian, Chao-Nan
;
Yan, Weiqun
;
Xing, Yanli
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2018/12/13
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
Xue, Xiaoqian
;
Zhang, Yan
;
Liu, Zhaoxuan
;
Song, Ming
;
Xing, Yanli
;
Xiang, Qiuping
;
Wang, Zhen
;
Tu, Zhengchao
;
Zhou, Yulai
;
Ding, Ke
;
Xu, Yong
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2016/12/16
The discovery of novel and selective fatty acid binding protein 4 inhibitors by virtual screening and biological evaluation
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 18, 页码: 4310-4317
Zhou, Yang
;
Nie, Tao
;
Zhang, Yan
;
Song, Ming
;
Li, Kuai
;
Ding, Mengxiao
;
Ding, Ke
;
Wu, Donghai
;
Xu, Yong
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2016/12/16
Identification of N-phenyl-2-(N-phenylphenylsulfonamido) acetamides as new ROR gamma inverse agonists: Virtual screening, structure-based optimization, and biological evaluation
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 116, 页码: 13-26
Song, Yu
;
Xue, Xiaoqian
;
Wu, Xishan
;
Wang, Rui
;
Xing, Yanli
;
Yan, Weiqun
;
Zhou, Yulai
;
Qian, Chao-Nan
;
Zhang, Yan
;
Xu, Yong
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2016/12/16
Discovery of 2-oxo-1,2-dihydrobenzo[cd]indole-6-sulfonamide derivatives as new ROR gamma inhibitors using virtual screening, synthesis and biological evaluation
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2014, 卷号: 78, 页码: 431-441
作者:
Zhang, Yan
;
Xue, Xiaoqian
;
Jin, Xiangyu
;
Song, Yu
;
Li, Jing
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2018/12/13
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