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科研机构
上海药物研究所 [59]
内容类型
期刊论文 [59]
发表日期
2020 [59]
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共59条,第1-10条
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发表日期:2020
专题:上海药物研究所
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A Peptide Binder of E3 Ligase Adaptor SPOP Disrupts Oncogenic SPOP-Protein Interactions in Kidney Cancer Cells
期刊论文
CHINESE JOURNAL OF CHEMISTRY, 2020, 页码: 274-280
作者:
Wang, Zhen
;
Zhang, Hao
;
Chen, Baoen
;
Ouyang, Sisheng
;
Zheng, Tong
收藏
  |  
浏览/下载:124/0
  |  
提交时间:2021/05/24
SPOP
Protein‐
protein interaction
Clear cell Renal Cell Carcinomas
Crystal structure
Peptide inhibitor
Targeted Proteomics Combined with Affinity Mass Spectrometry Analysis Reveals Antagonist E7 Acts As an Intracellular Covalent Ligand of Orphan Receptor GPR52
期刊论文
ACS CHEMICAL BIOLOGY, 2020, 卷号: 15, 期号: 12, 页码: 3275-3284
作者:
Ma, Mengna
;
Guo, Shimeng
;
Lin, Xi
;
Li, Shanshan
;
Wu, Yiran
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2021/05/24
A novel salviadione derivative, compound 15a, attenuates diabetes-induced renal injury by inhibiting NF-kappa B-mediated inflammatory responses
期刊论文
TOXICOLOGY AND APPLIED PHARMACOLOGY, 2020, 卷号: 409, 页码: 11
作者:
Li, Li
;
Ding, Chunyong
;
Zou, Chunpeng
;
Xiong, Zhi
;
Zhu, Weiwei
收藏
  |  
浏览/下载:98/0
  |  
提交时间:2021/05/24
Salviadione derivative 15a
Diabetic nephropathy
Inflammation
Macrophage infiltration
Fibrosis
Nuclear factor-kappa B
Cytokines
Diphyllin Improves High-Fat Diet-Induced Obesity in Mice Through Brown and Beige Adipocytes
期刊论文
FRONTIERS IN ENDOCRINOLOGY, 2020, 卷号: 11, 页码: 13
作者:
Duan, Ya-Nan
;
Ge, Xiang
;
Jiang, Hao-Wen
;
Zhang, Hong-Jie
;
Zhao, Yu
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2021/05/24
diphyllin
obesity
brown adipocyte
differentiation
thermogenesis
V-ATPase
Small molecules targeting the innate immune cGAS-STING-TBK1 signaling pathway
期刊论文
ACTA PHARMACEUTICA SINICA B, 2020, 卷号: 10, 期号: 12, 页码: 2272-2298
作者:
Ding, Chunyong
;
Song, Zilan
;
Shen, Ancheng
;
Chen, Tingting
;
Zhang, Ao
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2021/05/24
Immunotherapy
Anti-tumor
cGAS
STING
TBK1
Small molecule modulators
The Active Constituent From Gynostemma Pentaphyllum Prevents Liver Fibrosis Through Regulation of the TGF-beta 1/NDRG2/MAPK Axis
期刊论文
FRONTIERS IN GENETICS, 2020, 卷号: 11, 页码: 11
作者:
Huang, Hui
;
Wang, Kuifeng
;
Liu, Qian
;
Ji, Feihong
;
Zhou, Hu
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2020/12/24
HSC
TGF-β
1
liver fibrosis
quantitative proteomics
NDRG2
The novel small-molecule TPN10456 inhibits Th17 cell differentiation and protects against experimental autoimmune encephalomyelitis
期刊论文
CELLULAR & MOLECULAR IMMUNOLOGY, 2020, 页码: 4
作者:
Yang, Cuixia
;
Lv, Jie
;
Jiang, Xiangrui
;
Xiang, Zhenglong
;
Gong, Ran
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2020/12/24
Three dimensional drift control at nano-scale in single molecule localization microscopy
期刊论文
OPTICS EXPRESS, 2020, 卷号: 28, 期号: 22, 页码: 32750-32763
作者:
Fan, Xiaoming
;
Gensch, Thomas
;
Buldt, Georg
;
Zhang, Yuanheng
;
Musha, Zulipali
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2021/05/24
Engineering Prodrug Nanomedicine for Cancer Immunotherapy
期刊论文
ADVANCED SCIENCE, 2020, 页码: 33
作者:
Yang, Bin
;
Gao, Jing
;
Pei, Qing
;
Xu, Huixiong
;
Yu, Haijun
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2020/12/21
cancer immunotherapy
combination immunotherapy
nanomedicine
prodrugs
stimuli‐
responsive
A novel pectin from Polygala tenuifolia blocks A beta(42) aggregation and production by enhancing insulin-degradation enzyme and neprilysin
期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2020, 卷号: 161, 页码: 35-43
作者:
Zeng, Hui
;
Li, Piaopiao
;
Zhou, Lishuang
;
Ding, Kan
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2020/12/21
Polygala tenuifolia
Pectin
Polysaccharide
A beta(42) Alzheimer's disease
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