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THIAZOLO-PYRIMIDINE HIV-1 REVERSE TRANSCRIPTASE INHIBITOR, PREPARATION METHOD THEREFOR, AND USES THEREOF 专利
申请日期: 2019-10-17, 公开日期: 2019-10-17
作者:  Liu XY(刘新泳);  Kang DW(康东伟);  Zhan P(展鹏);  Wang Z(汪昭);  Wu GS(武高禅)
收藏  |  浏览/下载:34/0  |  提交时间:2020/01/04
FIVE-MEMBERED NON AROMATIC RING-PYRIMIDINE HIV-1 REVERSE TRANSCRIPTASE INHIBITOR, PREPARATION METHOD THEREFOR, AND USES THEREOF 专利
申请日期: 2019-10-17, 公开日期: 2019-10-17
作者:  Liu XY(刘新泳);  Kang DW(康东伟);  Zhan P(展鹏);  Wu GS(武高禅);  Wang Z(汪昭)
收藏  |  浏览/下载:26/0  |  提交时间:2020/01/04
Molecular Mechanism of Binding Selectivity of Inhibitors toward BACE1 and BACE2 Revealed by Multiple Short Molecular Dynamics Simulations and Free-Energy Predictions 期刊论文
ACS CHEMICAL NEUROSCIENCE, 2019, 卷号: 10, 期号: 10, 页码: 4303-4318
作者:  Chen, Jianzhong;  Wang, Jinan;  Yin, Baohua;  Pang, Laixue;  Wang, Wei
收藏  |  浏览/下载:114/0  |  提交时间:2020/07/01
Peptide self-assembly nanoparticles loaded with panobinostat to activate latent human immunodeficiency virus 期刊论文
Journal of biomedical nanotechnology, 2019, 卷号: 15, 期号: 5, 页码: 979-992
作者:  Kuai, Qiyuan;  Wang, Yu;  Gao, Fenghua;  Qi, Yingqiu;  Wang, Rui
收藏  |  浏览/下载:107/0  |  提交时间:2019/04/22
Peptide self-assembly nanoparticles loaded with panobinostat to activate latent human immunodeficiency virus 期刊论文
Journal of biomedical nanotechnology, 2019, 卷号: 15, 期号: 5, 页码: 979-992
作者:  Kuai, Qiyuan;  Wang, Yu;  Gao, Fenghua;  Qi, Yingqiu;  Wang, Rui
收藏  |  浏览/下载:107/0  |  提交时间:2019/04/22
Revisiting the mechanism of enfuvirtide and designing an analog with improved fusion inhibitory activity by targeting triple sites in gp41 期刊论文
AIDS, 2019, 卷号: 33, 期号: 10
作者:  Xu, Wei;  Pu, Jing;  Su, Shan;  Hua, Chen;  Su, Xiaojie
收藏  |  浏览/下载:19/0  |  提交时间:2019/12/05
Recent progress in HIV-1 inhibitors targeting the entrance channel of HIV-1 non-nucleoside reverse transcriptase inhibitor binding pocket 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 174
作者:  Gu, Shuang-Xi;  Xiao, Ting;  Zhu, Yuan-Yuan;  Liu, Gen-Yan;  Chen, Fen-Er
收藏  |  浏览/下载:11/0  |  提交时间:2019/12/05
A Peptide-Based HIV-1 Fusion Inhibitor with Two Tail-Anchors and Palmitic Acid Exhibits Substantially Improved In Vitro and Ex Vivo Anti-HIV-1 Activity and Prolonged In Vivo Half-Life 期刊论文
MOLECULES, 2019, 卷号: 24, 期号: 6
作者:  Su, Shan;  Rasquinha, Giselle;  Du, Lanying;  Wang, Qian;  Xu, Wei
收藏  |  浏览/下载:39/0  |  提交时间:2019/12/05
Development of Protein- and Peptide-Based HIV Entry Inhibitors Targeting gp120 or gp41 期刊论文
VIRUSES-BASEL, 2019, 卷号: 11, 期号: 8
作者:  Pu, Jing;  Wang, Qian;  Xu, Wei;  Lu, Lu;  Jiang, Shibo
收藏  |  浏览/下载:16/0  |  提交时间:2019/12/05
N-Substituted Pyrrole Derivative 12m Inhibits HIV-1 Entry by Targeting Gp41 of HIV-1 Envelope Glycoprotein 期刊论文
FRONTIERS IN PHARMACOLOGY, 2019, 卷号: 10
作者:  Qiu, Jiayin;  Liang, Taizhen;  Wu, Junyan;  Yu, Fei;  He, Xiaoyang
收藏  |  浏览/下载:18/0  |  提交时间:2019/12/05


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