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Disulfiram Copper Nanoparticles Prepared with a Stabilized Metal Ion Ligand Complex Method for Treating Drug-Resistant Prostate Cancers 期刊论文
ACS APPLIED MATERIALS & INTERFACES, 2018, 卷号: 10, 期号: 48, 页码: 41118-41128
作者:  Chen, Wu;  Yang, Wen;  Chen, Pengyu;  Huang, Yongzhuo;  Li, Feng
收藏  |  浏览/下载:96/0  |  提交时间:2019/01/08
Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants including T315I for chronic myeloid leukemia 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 160, 页码: 61-81
作者:  Liu, Xuesong;  Wang, Beilei;  Chen, Cheng;  Jiang, Zongru;  Hu, Chen
收藏  |  浏览/下载:14/0  |  提交时间:2019/01/11
A new class of HIV-1 inhibitors and the target identification via proteomic profiling 期刊论文
SCIENCE CHINA-CHEMISTRY, 2018, 卷号: 61, 期号: 11, 页码: 1430-1439
作者:  Ge, Ying-Zi;  Zhou, Bin;  Xiao, Ruo-Xuan;  Yuan, Xiao-Jing;  Zhou, Hu
收藏  |  浏览/下载:183/0  |  提交时间:2019/01/08
Synthesis of androgen receptor antagonists containing a pentafluorosulfanyl (SF5) moiety 期刊论文
ARCHIV DER PHARMAZIE, 2018, 卷号: 351, 期号: 11
作者:  Jin, Jiyu;  Zhou, Yan;  Yang, Dehua;  Zhang, Qiumeng;  Wang, Ming-Wei
收藏  |  浏览/下载:71/0  |  提交时间:2019/01/08
STAT3 activation confers trastuzumab-emtansine (T-DM1) resistance in HER2-positive breast cancer 期刊论文
CANCER SCIENCE, 2018, 卷号: 109, 期号: 10, 页码: 3305-3315
作者:  Wang, Lei;  Wang, Quanren;  Gao, Mingzhao;  Fu, Li;  Li, Yun
收藏  |  浏览/下载:51/0  |  提交时间:2019/01/08
Arsenic circumvents the gefitinib resistance by binding to P62 and mediating autophagic degradation of EGFR in non-small cell lung cancer 期刊论文
CELL DEATH & DISEASE, 2018, 卷号: 9
作者:  Mao, Jianhua;  Ma, Lie;  Shen, Yan;  Zhu, Kongkai;  Zhang, Ru
收藏  |  浏览/下载:49/0  |  提交时间:2019/01/08
Discovery of QCA570 as an Exceptionally Potent and Efficacious Proteolysis Targeting Chimera (PROTAC) Degrader of the Bromodomain and Extra-Terminal (BET) Proteins Capable of Inducing Complete and Durable Tumor Regression 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 15, 页码: 6685-6704
作者:  Qin, Chong;  Hu, Yang;  Zhou, Bing;  Fernandez-Salas, Ester;  Yang, Chao-Yie
收藏  |  浏览/下载:45/0  |  提交时间:2019/01/08
Synthesis and biological evaluation of novel larotaxel analogues 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 156, 页码: 692-710
作者:  Ren, Sumei;  Wang, Yujie;  Wang, Junfei;  Gao, Dingding;  Zhang, Minmin
收藏  |  浏览/下载:27/0  |  提交时间:2019/01/08
Screening and Identification of Lassa Virus Entry Inhibitors from an FDA-Approved Drug Library 期刊论文
JOURNAL OF VIROLOGY, 2018, 卷号: 92, 期号: 16, 页码: 14
作者:  Xiao, Gengfu;  Wang, Wei;  Liu, Yang;  Zhang, Guangshun;  Wang, Shaobo
收藏  |  浏览/下载:71/0  |  提交时间:2018/12/29
Activity of the chimeric lysin clyr against common gram-positive oral microbes and its anticaries efficacy in rat models 期刊论文
Viruses-basel, 2018, 卷号: 10, 期号: 7, 页码: 13
作者:  Xu, Jingjing;  Yang, Hang
收藏  |  浏览/下载:108/0  |  提交时间:2019/05/08


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