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Microenvironmental pH-modified solid dispersions to enhance the dissolution and bioavailability of poorly water-soluble weakly basic GT0918, a developing anti-prostate cancer drug: Preparation, characterization and evaluation in vivo
Yang, Meiyan[1]; He, Shaolong[2]; Fan, Yunzhou[3]; Wang, Yuli[4]; Ge, Zhenzhong[5]; Shan, Li[6]; Gong, Wei[7]; Huang, Xiaoli[8]; Tong, Youzhi[9]; Gao, Chunsheng[10]
刊名INTERNATIONAL JOURNAL OF PHARMACEUTICS
2014
卷号475期号:1-2页码:97-109
关键词Solid dispersion Microenvironmental pH Acidifier Poorly water soluble drug Bioavailability
ISSN号0378-5173
DOIhttp://dx.doi.org/10.1016/j.ijpharm.2014.08.047
URL标识查看原文
收录类别SCI(E) ; PUBMED
WOS记录号WOS:000345299500010
内容类型期刊论文
URI标识http://www.corc.org.cn/handle/1471x/5220969
专题河南大学
作者单位1.[1]Beijing Inst Pharmacol & Toxicol, Dept Pharmaceut, Beijing 100850, Peoples R China.
2.[2]Beijing Inst Pharmacol & Toxicol, Dept Pharmaceut, Beijing 100850, Peoples R China.
3.Cent S Univ, Sch Pharm, Changsha 410013, Hunan, Peoples R China.
4.[3]Peking Univ, Sch Pharmaceut Sci, Beijing 100191, Peoples R China.
5.[4]Beijing Inst Pharmacol & Toxicol, Dept Pharmaceut, Beijing 100850, Peoples R China.
6.[5]Henan Univ, Pharmaceut Coll, Kaifeng 475004, Peoples R China.
7.[6]Beijing Inst Pharmacol & Toxicol, Dept Pharmaceut, Beijing 100850, Peoples R China.
8.[7]Beijing Inst Pharmacol & Toxicol, Dept Pharmaceut, Beijing 100850, Peoples R China.
9.[8]Beijing Inst Pharmacol & Toxicol, Dept Pharmaceut, Beijing 100850, Peoples R China.
10.Cent S Univ, Sch Pharm, Changsha 410013, Hunan, Peoples R China.
推荐引用方式
GB/T 7714
Yang, Meiyan[1],He, Shaolong[2],Fan, Yunzhou[3],et al. Microenvironmental pH-modified solid dispersions to enhance the dissolution and bioavailability of poorly water-soluble weakly basic GT0918, a developing anti-prostate cancer drug: Preparation, characterization and evaluation in vivo[J]. INTERNATIONAL JOURNAL OF PHARMACEUTICS,2014,475(1-2):97-109.
APA Yang, Meiyan[1].,He, Shaolong[2].,Fan, Yunzhou[3].,Wang, Yuli[4].,Ge, Zhenzhong[5].,...&Gao, Chunsheng[10].(2014).Microenvironmental pH-modified solid dispersions to enhance the dissolution and bioavailability of poorly water-soluble weakly basic GT0918, a developing anti-prostate cancer drug: Preparation, characterization and evaluation in vivo.INTERNATIONAL JOURNAL OF PHARMACEUTICS,475(1-2),97-109.
MLA Yang, Meiyan[1],et al."Microenvironmental pH-modified solid dispersions to enhance the dissolution and bioavailability of poorly water-soluble weakly basic GT0918, a developing anti-prostate cancer drug: Preparation, characterization and evaluation in vivo".INTERNATIONAL JOURNAL OF PHARMACEUTICS 475.1-2(2014):97-109.
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