Fused heterocycles bearing bridgehead nitrogen as potent HIV-1 NNRTIs. Part 3: Optimization of [1,2,4]triazolo[1,5-a]pyrimidine core via structure-based and physicochemical property-driven approaches | |
Huang, Boshi; Li, Cuicui; Chen, Wenmin; Liu, Tao; Yu, Mingyan; Fu, Lu; Sun, Yueyue; Liu, Huiqing; De Clercq, Erik; Pannecouque, Christoph | |
刊名 | European Journal of Medicinal Chemistry: Chimie Therapeutique |
2015 | |
页码 | 754-765 |
关键词 | Triazolopyrimidines Structure-based drug design Biological activity HIV-1 RT Physicochemical properties Molecular simulations |
URL标识 | 查看原文 |
内容类型 | 期刊论文 |
URI标识 | http://www.corc.org.cn/handle/1471x/4772266 |
专题 | 山东大学 |
作者单位 | 1.Shandong Univ, Sch Pharmaceut Sci, Dept Med Chem, Key Lab Chem Biol,Minist Educ, Jinan 250012 2.Shandong Univ, Sch Pharmaceut Sci |
推荐引用方式 GB/T 7714 | Huang, Boshi,Li, Cuicui,Chen, Wenmin,et al. Fused heterocycles bearing bridgehead nitrogen as potent HIV-1 NNRTIs. Part 3: Optimization of [1,2,4]triazolo[1,5-a]pyrimidine core via structure-based and physicochemical property-driven approaches[J]. European Journal of Medicinal Chemistry: Chimie Therapeutique,2015:754-765. |
APA | Huang, Boshi.,Li, Cuicui.,Chen, Wenmin.,Liu, Tao.,Yu, Mingyan.,...&Pannecouque, Christoph.(2015).Fused heterocycles bearing bridgehead nitrogen as potent HIV-1 NNRTIs. Part 3: Optimization of [1,2,4]triazolo[1,5-a]pyrimidine core via structure-based and physicochemical property-driven approaches.European Journal of Medicinal Chemistry: Chimie Therapeutique,754-765. |
MLA | Huang, Boshi,et al."Fused heterocycles bearing bridgehead nitrogen as potent HIV-1 NNRTIs. Part 3: Optimization of [1,2,4]triazolo[1,5-a]pyrimidine core via structure-based and physicochemical property-driven approaches".European Journal of Medicinal Chemistry: Chimie Therapeutique (2015):754-765. |
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