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Fused heterocycles bearing bridgehead nitrogen as potent HIV-1 NNRTIs. Part 3: Optimization of [1,2,4]triazolo[1,5-a]pyrimidine core via structure-based and physicochemical property-driven approaches
Huang, Boshi; Li, Cuicui; Chen, Wenmin; Liu, Tao; Yu, Mingyan; Fu, Lu; Sun, Yueyue; Liu, Huiqing; De Clercq, Erik; Pannecouque, Christoph
刊名European Journal of Medicinal Chemistry: Chimie Therapeutique
2015
页码754-765
关键词Triazolopyrimidines Structure-based drug design Biological activity HIV-1 RT Physicochemical properties Molecular simulations
URL标识查看原文
内容类型期刊论文
URI标识http://www.corc.org.cn/handle/1471x/4772266
专题山东大学
作者单位1.Shandong Univ, Sch Pharmaceut Sci, Dept Med Chem, Key Lab Chem Biol,Minist Educ, Jinan 250012
2.Shandong Univ, Sch Pharmaceut Sci
推荐引用方式
GB/T 7714
Huang, Boshi,Li, Cuicui,Chen, Wenmin,et al. Fused heterocycles bearing bridgehead nitrogen as potent HIV-1 NNRTIs. Part 3: Optimization of [1,2,4]triazolo[1,5-a]pyrimidine core via structure-based and physicochemical property-driven approaches[J]. European Journal of Medicinal Chemistry: Chimie Therapeutique,2015:754-765.
APA Huang, Boshi.,Li, Cuicui.,Chen, Wenmin.,Liu, Tao.,Yu, Mingyan.,...&Pannecouque, Christoph.(2015).Fused heterocycles bearing bridgehead nitrogen as potent HIV-1 NNRTIs. Part 3: Optimization of [1,2,4]triazolo[1,5-a]pyrimidine core via structure-based and physicochemical property-driven approaches.European Journal of Medicinal Chemistry: Chimie Therapeutique,754-765.
MLA Huang, Boshi,et al."Fused heterocycles bearing bridgehead nitrogen as potent HIV-1 NNRTIs. Part 3: Optimization of [1,2,4]triazolo[1,5-a]pyrimidine core via structure-based and physicochemical property-driven approaches".European Journal of Medicinal Chemistry: Chimie Therapeutique (2015):754-765.
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