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Discovery of 1,8-acridinedione derivatives as novel GCN5 inhibitors via high throughput screening
Xiong, Huan[1]; Han, Jie[2]; Wang, Jun[3]; Lu, Wenchao[4]; Wang, Chen[5]; Chen, Yu[6]; Lian, Fulin[7]; Zhang, Naixia[8]; Liu, Yu-Chih[9]; Zhang, Chenhua[10]
刊名EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
2018
卷号151页码:740-751
关键词Epigenetics Histone acetyltransferase GCN5 High throughput screening 1 8-Acridinedione derivative
ISSN号0223-5234
URL标识查看原文
内容类型期刊论文
URI标识http://www.corc.org.cn/handle/1471x/2181016
专题上海大学
作者单位1.[1]Shanghai Univ, Dept Chem, Coll Sci, 99 Shangda Rd, Shanghai 200444, Peoples R China.
2.Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China.
3.[2]Chinese Acad Sci, Shanghai Inst Mat Med, CAS Key Lab Receptor Res, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China.
4.[3]Chinese Acad Sci, Shanghai Inst Mat Med, CAS Key Lab Receptor Res, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China.
5.Nanjing Univ Chinese Med, Jiangsu Key Lab High Technol Res TCM Formulae, 138 Xianlin Rd, Nanjing 210023, Jiangsu, Peoples R China.
6.[4]Chinese Acad Sci, Shanghai Inst Mat Med, CAS Key Lab Receptor Res, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China.
7.Univ Chinese Acad Sci, 19 Yuquan Rd, Beijing 100049, Peoples R China.
8.[5]Chinese Acad Sci, Shanghai Inst Mat Med, CAS Key Lab Receptor Res, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China.
9.Univ Chinese Acad Sci, 19 Yuquan Rd, Beijing 100049, Peoples R China.
10.[6]Chinese Acad Sci, Shanghai Inst Mat Med, CAS Key Lab Receptor Res, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China.
推荐引用方式
GB/T 7714
Xiong, Huan[1],Han, Jie[2],Wang, Jun[3],et al. Discovery of 1,8-acridinedione derivatives as novel GCN5 inhibitors via high throughput screening[J]. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY,2018,151:740-751.
APA Xiong, Huan[1].,Han, Jie[2].,Wang, Jun[3].,Lu, Wenchao[4].,Wang, Chen[5].,...&Zhou, Bing[15].(2018).Discovery of 1,8-acridinedione derivatives as novel GCN5 inhibitors via high throughput screening.EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY,151,740-751.
MLA Xiong, Huan[1],et al."Discovery of 1,8-acridinedione derivatives as novel GCN5 inhibitors via high throughput screening".EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 151(2018):740-751.
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