Synthesis and Biological Activities of 1,2,3-Thiadiazole Derivatives Containing 1,3,4-Thiadiazole Moiety | |
Wang Shouxin1,2; Zuo Xiang2; Fan Zhijin2; Zhang Zhengcai2; Zhang Jufang2; Xiong Lixia2; Fu Yifeng2; Fang Zhen2; Wu Qingjun3; Zhang Youjun3 | |
刊名 | CHINESE JOURNAL OF ORGANIC CHEMISTRY |
2013 | |
卷号 | 33期号:11页码:2367-2375 |
关键词 | 1,2,3-thiadiazole 1,3,4-thiadiazole synthesis fungicidal activity insecticidal activity |
ISSN号 | 0253-2786 |
DOI | 10.6023/cjoc201306002 |
通讯作者 | Wang Shouxin |
英文摘要 | To find novel pesticide lead compounds with highly active bioactivity, 32 novel 1,2,3-thiadiazole derivatives containing 1,3,4-thiadiazole ring were designed and synthesized according to the principle of combination of bioactive substructures. All structures were confirmed by H-1 NMR, IR and HRMS. The fungicidal and insecticidal activities of these compounds were also evaluated. The bioassay results showed that some target compounds had good fungicidal activity and excellent insecticidal activities. Among them, compounds 5-3, 5-20 and 5-31 showed similar insecticidal activity against Plutella xylostella L. as compared with positive control chlorfluazuron at the same condition, compounds 5-6, 5-7, 5-10, 5-14 and 5-17 presented 100% insecticidal activity against Culex pipiens pollen at the concentration of 5 mu g/mL. |
学科主题 | Chemistry, Organic ; CHEMISTRY, ORGANIC |
语种 | 中文 |
出版者 | SCIENCE PRESS |
WOS记录号 | WOS:000328597700012 |
内容类型 | 期刊论文 |
源URL | [http://111.203.20.206/handle/2HMLN22E/101022] |
专题 | 蔬菜花卉研究所_职能部门 |
作者单位 | 1.Jining Med Univ, Sch Basic Sci, Jining 272067, Peoples R China 2.Nankai Univ, State Key Lab Elementoorgan Chem, Tianjin 300071, Peoples R China 3.Chinese Acad Agr Sci, Inst Vegetables & Flowers, Beijing 100081, Peoples R China |
推荐引用方式 GB/T 7714 | Wang Shouxin,Zuo Xiang,Fan Zhijin,et al. Synthesis and Biological Activities of 1,2,3-Thiadiazole Derivatives Containing 1,3,4-Thiadiazole Moiety[J]. CHINESE JOURNAL OF ORGANIC CHEMISTRY,2013,33(11):2367-2375. |
APA | Wang Shouxin.,Zuo Xiang.,Fan Zhijin.,Zhang Zhengcai.,Zhang Jufang.,...&Zhang Youjun.(2013).Synthesis and Biological Activities of 1,2,3-Thiadiazole Derivatives Containing 1,3,4-Thiadiazole Moiety.CHINESE JOURNAL OF ORGANIC CHEMISTRY,33(11),2367-2375. |
MLA | Wang Shouxin,et al."Synthesis and Biological Activities of 1,2,3-Thiadiazole Derivatives Containing 1,3,4-Thiadiazole Moiety".CHINESE JOURNAL OF ORGANIC CHEMISTRY 33.11(2013):2367-2375. |
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